Discoidin Domain Receptor Inhibitors

DDR1, IC₅₀: 29 nM

DDR2, IC₅₀: 0.5 nM

DDR2, IC₅₀: 230 nM

DDR1

DDR1, IC₅₀: 46.16 nM

DDR1, IC₅₀: 57 nM

DDR1, IC₅₀: 4.67 nM

DDR2, IC₅₀: 7.39 nM

DDR2, IC₅₀: 3.2 nM

DDR1, IC₅₀: 29 nM

DDR2, IC₅₀: 1900 nM

DDR1, IC₅₀: 9.72 nM

DDR1, IC₅₀: 7.36 nM

DDR1

DDR2

DDR1, IC₅₀: 29 nM

DDR2, IC₅₀: 0.5 nM

DDR2, IC₅₀: 7.0 nM

DDR1, IC₅₀: 23 nM

DDR2, IC₅₀: 18 nM

DDR2, IC₅₀: 6.105 μM

DDR1

DDR2

DDR1, IC₅₀: 9.4 nM

DDR2, IC₅₀: 20.4 nM

DDR1, IC₅₀: 105 nM

DDR2, IC₅₀: 413 nM